Artefenomel Regioisomer RLA-3107 Is a Promising Lead for the Discovery of Next-Generation Endoperoxide Antimalarials. Read more about Artefenomel Regioisomer RLA-3107 Is a Promising Lead for the Discovery of Next-Generation Endoperoxide Antimalarials.
Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers. Read more about Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers. Read more about Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
A Phosphoramidate Strategy Enables Membrane Permeability of a Non-nucleotide Inhibitor of the Prolyl Isomerase Pin1. Read more about A Phosphoramidate Strategy Enables Membrane Permeability of a Non-nucleotide Inhibitor of the Prolyl Isomerase Pin1.
Optimization of Phenyl Indole Inhibitors of the AAA+ ATPase p97. Read more about Optimization of Phenyl Indole Inhibitors of the AAA+ ATPase p97.
Exploring N-Arylsulfonyl-l-proline Scaffold as a Platform for Potent and Selective αvβ1 Integrin Inhibitors. Read more about Exploring N-Arylsulfonyl-l-proline Scaffold as a Platform for Potent and Selective αvβ1 Integrin Inhibitors.
Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway. Read more about Allosteric Indole Amide Inhibitors of p97: Identification of a Novel Probe of the Ubiquitin Pathway.
Structure-Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97. Read more about Structure-Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97.
Trioxolane-Mediated Delivery of Mefloquine Limits Brain Exposure in a Mouse Model of Malaria. Read more about Trioxolane-Mediated Delivery of Mefloquine Limits Brain Exposure in a Mouse Model of Malaria.
Development of novel Vitamin D Receptor-Coactivator Inhibitors. Read more about Development of novel Vitamin D Receptor-Coactivator Inhibitors.
