Predicting and improving the membrane permeability of peptidic small molecules. Read more about Predicting and improving the membrane permeability of peptidic small molecules.
Structure-based design of potent and ligand-efficient inhibitors of CTX-M class A β-lactamase. Read more about Structure-based design of potent and ligand-efficient inhibitors of CTX-M class A β-lactamase.
Investigating the antimalarial action of 1,2,4-trioxolanes with fluorescent chemical probes. Read more about Investigating the antimalarial action of 1,2,4-trioxolanes with fluorescent chemical probes.
Chemical structural novelty: on-targets and off-targets. Read more about Chemical structural novelty: on-targets and off-targets.
Profiling of a prescription drug library for potential renal drug-drug interactions mediated by the organic cation transporter 2. Read more about Profiling of a prescription drug library for potential renal drug-drug interactions mediated by the organic cation transporter 2.
Irreversible Nek2 kinase inhibitors with cellular activity. Read more about Irreversible Nek2 kinase inhibitors with cellular activity.
2-Aminothiazoles as therapeutic leads for prion diseases. Read more about 2-Aminothiazoles as therapeutic leads for prion diseases.
Heat shock protein 70 (hsp70) as an emerging drug target. Read more about Heat shock protein 70 (hsp70) as an emerging drug target.
Molecular shape and medicinal chemistry: a perspective. Read more about Molecular shape and medicinal chemistry: a perspective.
Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB. Read more about Identification and optimization of inhibitors of Trypanosomal cysteine proteases: cruzain, rhodesain, and TbCatB.