How This Cancer Drug Could Make Radiation a Slam Dunk Therapy

UCSF scientists combine a precision drug therapy with an antibody and radiation to eliminate tumors without causing side effects.

By Levi Gadye | UCSF.edu | December 10, 2024

A 3D rendering showing immune proteins delivering K R A S, and others a radioactive antibody, to a tumor cell.

Radiation is one of the most effective ways to kill a tumor. But these therapies are indiscriminate, and they can damage healthy tissues.

Now, UC San Francisco scientists have developed a way to deliver radiation just to cancerous cells. The therapy combines a drug to mark the cancer cells for destruction and a radioactive antibody to kill them.

It wiped out bladder and lung tumors in mice without causing lethargy or weight loss – the typical side effects of radiation therapy.

“This is a one-two punch,” said Charly Craik, PhD, a professor of pharmaceutical chemistry at UCSF and co-senior author of the study, which appears Dec. 10 in Cancer Research. “We could potentially kill the tumors before they can develop resistance.”

A cancer drug becomes a molecular flag for cancer

The project began 10 years ago when UCSF’s Kevan Shokat, PhD, discovered how to attack KRAS, a notorious cancer-causing protein. When mutated, KRAS spurs out-of-control cell growth. Such mutations lead to up to a third of all cancer.

Read more at UCSF.edu