Systematic Study of Heteroarene Stacking Using a Congeneric Set of Molecular Glues for Procaspase-6. Read more about Systematic Study of Heteroarene Stacking Using a Congeneric Set of Molecular Glues for Procaspase-6.
Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes. Read more about Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes.
First-in-Class Allosteric Inhibitors of DNMT3A Disrupt Protein-Protein Interactions and Induce Acute Myeloid Leukemia Cell Differentiation. Read more about First-in-Class Allosteric Inhibitors of DNMT3A Disrupt Protein-Protein Interactions and Induce Acute Myeloid Leukemia Cell Differentiation.
Drugging the Next Undruggable KRAS Allele-Gly12Asp. Read more about Drugging the Next Undruggable KRAS Allele-Gly12Asp.
Colloidal Aggregators in Biochemical SARS-CoV-2 Repurposing Screens. Read more about Colloidal Aggregators in Biochemical SARS-CoV-2 Repurposing Screens.
Inhibitor Combinations Reveal Wiring of the Proteostasis Network in Prostate Cancer Cells. Read more about Inhibitor Combinations Reveal Wiring of the Proteostasis Network in Prostate Cancer Cells.
Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery. Read more about Re-emerging Aspartic Protease Targets: Examining Cryptococcus neoformans Major Aspartyl Peptidase 1 as a Target for Antifungal Drug Discovery.
Conformational Strain of Macrocyclic Peptides in Ligand-Receptor Complexes Based on Advanced Refinement of Bound-State Conformers. Read more about Conformational Strain of Macrocyclic Peptides in Ligand-Receptor Complexes Based on Advanced Refinement of Bound-State Conformers.
XGen: Real-Space Fitting of Complex Ligand Conformational Ensembles to X-ray Electron Density Maps. Read more about XGen: Real-Space Fitting of Complex Ligand Conformational Ensembles to X-ray Electron Density Maps.
Fragment-based Differential Targeting of PPI Stabilizer Interfaces. Read more about Fragment-based Differential Targeting of PPI Stabilizer Interfaces.