Large Library Docking and Biophysical Analysis of Small-Molecule TMPRSS2 Inhibitors. Read more about Large Library Docking and Biophysical Analysis of Small-Molecule TMPRSS2 Inhibitors.
Promise and Challenge of β-Lactone Electrophiles to Target Aspartate 12 of Mutant KRASG12D. Read more about Promise and Challenge of β-Lactone Electrophiles to Target Aspartate 12 of Mutant KRASG12D.
On-Resin Assembly of Macrocyclic Inhibitors of Cryptococcus neoformans May1: A Pathway to Potent Antifungal Agents. Read more about On-Resin Assembly of Macrocyclic Inhibitors of Cryptococcus neoformans May1: A Pathway to Potent Antifungal Agents.
Overcoming Secondary Mutations of Type II Kinase Inhibitors. Read more about Overcoming Secondary Mutations of Type II Kinase Inhibitors.
Systematic Study of Heteroarene Stacking Using a Congeneric Set of Molecular Glues for Procaspase-6. Read more about Systematic Study of Heteroarene Stacking Using a Congeneric Set of Molecular Glues for Procaspase-6.
Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes. Read more about Development and Characterization of Type I, Type II, and Type III LIM-Kinase Chemical Probes.
First-in-Class Allosteric Inhibitors of DNMT3A Disrupt Protein-Protein Interactions and Induce Acute Myeloid Leukemia Cell Differentiation. Read more about First-in-Class Allosteric Inhibitors of DNMT3A Disrupt Protein-Protein Interactions and Induce Acute Myeloid Leukemia Cell Differentiation.
Drugging the Next Undruggable KRAS Allele-Gly12Asp. Read more about Drugging the Next Undruggable KRAS Allele-Gly12Asp.
Colloidal Aggregators in Biochemical SARS-CoV-2 Repurposing Screens. Read more about Colloidal Aggregators in Biochemical SARS-CoV-2 Repurposing Screens.
Inhibitor Combinations Reveal Wiring of the Proteostasis Network in Prostate Cancer Cells. Read more about Inhibitor Combinations Reveal Wiring of the Proteostasis Network in Prostate Cancer Cells.
